Items where Author is "Docsa, Tibor"

Article

Nagy, Lilla Nikoletta and Márton, Judit and Vida, András and Kis, G. and Bokor, Éva and Kun, Sándor and Docsa, Tibor and Gergely, Pál and Pacher, Pál and Somsák, László and Bay, Péter (2017) Glycogen phosphorylase inhibition improves β-cell function. BRITISH JOURNAL OF PHARMACOLOGY. pp. 1-19. ISSN 0007-1188

Donnier-Maréchal, Marion and Goyard, David and Folliard, Vincent and Docsa, Tibor and Gergely, Pál and Praly, Jean-Pierre and Vidal, Sébastien (2015) 3-Glucosylated 5-amino-1,2,4-oxadiazoles : synthesis and evaluation as glycogen phosphorylase inhibitors. BEILSTEIN JOURNAL OF ORGANIC CHEMISTRY, 11. pp. 499-503. ISSN 1860-5397

Bokor, Éva and Szennyes, Eszter and Csupász, Tibor and Tóth, Nóra and Docsa, Tibor and Gergely, Pál and Somsák, László (2015) C-(2-Deoxy-D-arabino-hex-1-enopyranosyl)-oxadiazoles: synthesis of possible isomers and their evaluation as glycogen phosphorylase inhibitors. Carbohydrate Research, 412. pp. 71-79. ISSN 0008-6215

Begum, J. and Varga, G. and Docsa, Tibor and Gergely, Pál and Hayes, J. M. and Juhász, László and Somsák, László (2015) Computationally motivated synthesis and enzyme kinetic evaluation of N-(β-D-glucopyranosyl)-1,2,4-triazolecarboxamides as glycogen phosphorylase inhibitors. MEDCHEMCOMM, 6. pp. 80-89. ISSN 2040-2503

Docsa, Tibor and Marics, B. and Németh, J. and Hüse, Cs. and Somsák, L. and Gergely, Pál (2015) Insulin sensitivity is modified by a glycogen phosphorylase inhibitor: glucopyranosylidene-spiro-thiohydantoin in streptozotocin-induced diabetic rats. CURRENT TOPICS IN MEDICINAL CHEMISTRY, 15. pp. 1-5. ISSN 1568-0266

Goyard, D. and Docsa, Tibor and Gergely, Pál and Praly, J-P. and Vidal, S. (2015) Synthesis of 4-amidomethyl-1-glucosyl-1,2,3-triazoles and evaluation as glycogen phosphorylase inhibitors. CARBOHYDRATE RESEARCH, 402. pp. 245-251. ISSN 0008-6215

Czifrák, Katalin and Páhi, A. and Deák, Sz. and Kiss, Attila and E Kövér, Katalin and Docsa, Tibor and Gergely, Pál and Somsák, László (2014) Glucopyranosylidene-spiro-iminothiazolidinone, a new bicyclic ring system: synthesis, derivatization, and evaluation for inhibition of glycogen phosphorylase by enzyme kinetic and crystallographic methods. BIOORGANIC & MEDICINAL CHEMISTRY, 22. pp. 4028-4041. ISSN 0968-0896

Kun, Sándor and Bokor, Éva and Varga, G. and Szőcs, B. and Páhi, A. and Vágvölgyiné Tóth, Marietta and Juhász, László and Docsa, Tibor and Gergely, Pál and Somsák, László (2014) New synthesis of 3-(beta-D-glucopyranosyl)-5-substituted-1,2,4-triazoles, nanomolar inhibitors of glycogen phosphorylase. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 76. pp. 567-579. ISSN 0223-5234

Juhász, László and Varga, G. and Sztankovics, A. and Béke, F. and Docsa, Tibor and Kiss, Attila and Gergely, Pál and Somsák, László (2014) Structure-activity relationships of glycogen phosphorylase inhibitor FR258900 and its analogues: a combined synthetic, enzyme kinetics, and computational study. CHEMPLUSCHEM, 79 (11). pp. 1558-1568. ISSN 2192-6506

Somsák, László and Bokor, Éva and Czibere, B. and Czifrák, Katalin and Koppány, Cs. and Kun, Sándor and Vágvölgyiné Tóth, Marietta and Docsa, Tibor and Gergely, Pál (2014) Synthesis of C-xylopyranosyl- and xylopyranosylidene-spiro-heterocycles as potential inhibitors of glycogen phosphorylase. Carbohydrate Research, 399. pp. 38-48. ISSN 0008-6215

Varga, Gergely and Docsa, Tibor and Gergely, Pál and Juhász, László and Somsák, László (2013) Synthesis of tartaric acid analogues of FR258900 and their evaluation as glycogen phosphorylase inhibitors. Bioorganic & medicinal chemistry letters, 23 (6). pp. 1789-92. ISSN 1464-3405

Bokor, Éva and Docsa, Tibor and Gergely, Pál and Somsák, László (2013) C-Glucopyranosyl-1,2,4-triazoles As New Potent Inhibitors of Glycogen Phosphorylase. ACS MEDICINAL CHEMISTRY LETTERS, 4 (7). pp. 612-615. ISSN 1948-5875

Nagy, Lilla Nikoletta and Docsa, Tibor and Brunyánszki, Attila and Szántó, Magdolna and Hegedűs, Csaba and Márton, Judit and Virág, László and Somsák, László and Gergely, Pál and Bay, Péter (2013) Glycogen phosphorylase inhibitor N-(3,5-dimethyl-benzoyl)-N'-(β-Dglucopyranosyl) urea improves glucose tolerance under normoglycemic and diabetic conditions and rearranges hepatic metabolism. PLOS ONE, 8 (7). e69420. ISSN 1932-6203

Tóth, Marietta and Szőcs, Béla and Kaszás, Tímea and Docsa, Tibor and Gergely, Pál and Somsák, László (2013) Synthesis of 2-(β-D-glucopyranosylamino)-5-substituted-1,3,4-oxadiazoles for inhibition of glycogen phosphorylase. CARBOHYDRATE RESEARCH, 381. pp. 196-204. ISSN 0008-6215

Szőcs, Béla and Tóth, Marietta and Docsa, Tibor and Gergely, Pál and Somsák, László (2013) Synthesis of 2-(β-d-glucopyranosyl)-5-(substituted-amino)-1,3,4-oxa- and -thiadiazoles for the inhibition of glycogen phosphorylase. CARBOHYDRATE RESEARCH, 381. pp. 187-195. ISSN 0008-6215

Bokor, Éva and Szilágyi, Enikő and Docsa, Tibor and Gergely, Pál and Somsák, László (2013) Synthesis of substituted 2-(β-d-glucopyranosyl)-benzimidazoles and their evaluation as inhibitors of glycogen phosphorylase. Carbohydrate Research, 381. pp. 179-186. ISSN 0008-6215

Varga, G. and Docsa, Tibor and Gergely, Pál and Juhász, László and Somsák, László (2013) Synthesis of tartaric acid analogues of FR258900 and their evaluation as glycogen phosphorylase inhibitors. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 23. pp. 1789-1792. ISSN 0960-894X

Polyák, M. and Varga, G. and Szilágyi, Bence and Juhász, László and Docsa, Tibor and Gergely, Pál and Somsák, László (2013) Synthesis, enzyme kinetics and computational evaluation of N-(beta-D-glucopyranosyl) oxadiazolecarboxamides as glycogen phosphorylase inhibitors. BIOORGANIC & MEDICINAL CHEMISTRY, 21. pp. 5738-5747. ISSN 0968-0896