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Items where Author is "Jójárt, Rebeka"

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Number of items: 13.

Article

Mernyák, Erzsébet and Bartha, Sándor and Kóczán, Lili and Jójárt, Rebeka and Resch, Vivien and Paragi, Gábor and Vágvölgyi, Máté and Hunyadi, Attila and Bruszel, Bella and Zupkó, István and Minorics, Renáta (2021) Microwave-assisted Phospha-Michael addition reactions in the 13α-oestrone series and in vitro antiproliferative properties. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 36 (1). pp. 1931-1937. ISSN 1475-6366

Sinreih, Masa and Jójárt, Rebeka and Kele, Zoltán and Budefeld, Tomaz and Paragi, Gábor and Mernyák, Erzsébet and Lanisnik-Rizner, Tea (2021) Synthesis and evaluation of AKR1C inhibitory properties of A-ring halogenated oestrone derivatives. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 36 (1). pp. 1500-1508. ISSN 1475-6366

Laczkó-Rigó, Réka and Bakos, Éva and Jójárt, Rebeka and Tömböly, Csaba and Mernyák, Erzsébet and Özvegy-Laczka, Csilla (2021) Selective antiproliferative effect of C-2 halogenated 13α-estrones on cells expressing Organic anion-transporting polypeptide 2B1 (OATP2B1). TOXICOLOGY AND APPLIED PHARMACOLOGY. ISSN 0041-008X

Kiss, Anita and Jójárt, Rebeka and Mernyák, Erzsébet and Bartha, Sándor and Minorics, Renáta and Zupkó, István and Schneider, Gyula (2021) Novel preparation of substituted oxazolines condensed to d-ring of estrane skeleton and characterization of their antiproliferative properties. STEROIDS. ISSN 0039-128X (In Press)

Jójárt, Rebeka and Laczkó-Rigó, Réka and Klement, Máté and Kőhl, Gabriella and Kecskeméti, Gábor and Laczka, Csilla and Mernyák, Erzsébet (2021) Design, synthesis and biological evaluation of novel estrone phosphonates as high affinity organic anion-transporting polypeptide 2B1 (OATP2B1) inhibitors. BIOORGANIC CHEMISTRY. ISSN 0045-2068 (Unpublished)

Sinreih, Maša and Jójárt, Rebeka and Kele, Zoltán and Büdefeld, Tomaž and Paragi, Gábor and Mernyák, Erzsébet (2021) Synthesis and evaluation of AKR1C inhibitory properties of A-ring halogenated oestrone derivatives. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 36 (1). pp. 1500-1508. ISSN 1475-6366

Jójárt, Rebeka and Senobar Tahaei, Seyyed Ashkan and Trungel-Nagy, Péter and Kele, Zoltán and Minorics, Renáta and Paragi, Gábor and Zupkó, István and Mernyák, Erzsébet (2021) Synthesis and evaluation of anticancer activities of 2- or 4-substituted 3-(N-benzyltriazolylmethyl)-13α-oestrone derivatives. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 36 (1). pp. 58-67. ISSN 1475-6366

Jójárt, Rebeka and Ali, Hazhmat and Horváth, Gergely and Kele, Zoltán and Zupkó, István and Mernyák, Erzsébet (2020) Pd-Catalyzed Suzuki–Miyaura couplings and evaluation of 13α-estrone derivatives as potential anticancer agents. STEROIDS, 164. ISSN 0039-128X

Laczkó-Rigó, Réka and Jójárt, Rebeka and Mernyák, Erzsébet and Bakos, Éva and Tuerkova, Alzbeta and Özvegy-Laczka, Csilla (2020) Structural dissection of 13-epiestrones based on the interaction with human Organic anion-transporting polypeptide, OATP2B1. JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 200. pp. 1-10. ISSN 0960-0760

Jójárt, Rebeka and Traj, Péter and Kovács, Édua and Horváth, Ágnes and Schneider, Gyula and Szécsi, Mihály and Pál, Attila and Paragi, Gábor and Mernyák, Erzsébet (2019) Synthesis, Biological Evaluation and Docking Studies of 13-Epimeric 10-fluoro- and 10-Chloroestra-1,4-dien-3-ones as Potential Aromatase Inhibitors. MOLECULES, 24 (9). No.-1783. ISSN 1420-3049

Jójárt, Rebeka and Pécsy, Balázs and Keglevich, György and Szécsi, Mihály and Rigó, Réka and Laczka, Csilla and Mernyák, Erzsébet (2018) Pd-Catalyzed microwave-assisted synthesis of phosphonated 13α-estrones as potential OATP2B1, 17β-HSD1 and/or STS inhibitors. BEILSTEIN JOURNAL OF ORGANIC CHEMISTRY, 14. pp. 2838-2845. ISSN 1860-5397

Bacsa, Ildikó and Herman, Bianka Edina and Jójárt, Rebeka and Herman, Kevin Stefán and Wölfling, János and Schneider, Gyula and Varga, Mónika and Tömböly, Csaba and Szécsi, Mihály and Mernyák, Erzsébet (2018) Synthesis and structure–activity relationships of 2- and/or 4-halogenated 13β- and 13α-estrone derivatives as enzyme inhibitors of estrogen biosynthesis. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 33 (1). pp. 1271-1282. ISSN 1475-6366 (print); 1475-6374 (online)

Bacsa, Ildikó and Jójárt, Rebeka and Wölfling, János and Schneider, Gyula and Herman, Bianka Edina and Szécsi, Mihály and Mernyák, Erzsébet (2017) Synthesis of novel 13 α-estrone derivatives by Sonogashira coupling as potential 17 β-HSD1 inhibitors. BEILSTEIN JOURNAL OF ORGANIC CHEMISTRY, 13. pp. 1303-1309. ISSN 1860-5397

This list was generated on Fri Mar 29 16:36:33 2024 CET.