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Items where Author is "Tömböly, Csaba"

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Number of items: 43.

Dvorácskó, Szabolcs and Körmöczi, Tímea and Sija, Éva and Bende, Balázs and Weiczner, Roland and Varga, Tibor and Ilisz, István and Institóris, László and Kereszty, Éva M. and Tömböly, Csaba and Berkecz, Róbert (2023) Focusing on the 5F-MDMB-PICA, 4F-MDMB-BICA Synthetic Cannabinoids and Their Primary Metabolites in Analytical and Pharmacological Aspects. TOXICOLOGY AND APPLIED PHARMACOLOGY, 470. No.-116548. ISSN 0041-008X (print); 1096-0333 (online)

Dvorácskó, Szabolcs and Dimmito, Marilisa Pia and Sebastiani, Jessica and La Regina, Giuseppe and Silvestri, Romano and Tömböly, Csaba (2023) Rimonabant-Based Compounds Bearing Hydrophobic Amino Acid Derivatives as Cannabinoid Receptor Subtype 1 Ligands. ACS MEDICINAL CHEMISTRY LETTERS, 14 (4). pp. 479-486. ISSN 1948-5875

Bauder-Wuest, Ulrike and Schaefer, Martin and Winter, Ruth and Remde, Yvonne and Roscher, Mareike and Breyl, Heinz and Poethko, Thorsten and Tömböly, Csaba and Benešová-Schäfer, Martina (2023) Synthesis of tritium-labeled Lu-PSMA-617: Alternative tool for biological evaluation of radiometal-based pharmaceuticals. APPLIED RADIATION AND ISOTOPES, 197. No-110819. ISSN 0969-8043

Laczkó-Rigó, Réka and Bakos, Éva and Jójárt, Rebeka and Tömböly, Csaba and Mernyák, Erzsébet and Özvegy-Laczka, Csilla (2021) Selective antiproliferative effect of C-2 halogenated 13α-estrones on cells expressing Organic anion-transporting polypeptide 2B1 (OATP2B1). TOXICOLOGY AND APPLIED PHARMACOLOGY. ISSN 0041-008X

Hus-Citharel, Annette and Bouby, Nadine and Corbani, Maithé and Mion, Julie and Mendre, Christiane and Darusi, Judit and Tömböly, Csaba (2021) Characterization of a Functional V1B Vasopressin Receptor in the Male Rat Kidney: Evidence for Cross Talk Between V1B and V2 Receptor Signaling Pathways. AMERICAN JOURNAL OF PHYSIOLOGY - RENAL PHYSIOLOGY, 321 (3). pp. 305-321. ISSN 1931-857X (print); 1522-1466 (online)

Almási, Nikoletta and Murlasits, Z. and Al-Awar, Amin and Csonka, Ákos and Dvorácskó, Szabolcs and Tömböly, Csaba and Török, Szilvia and Pósa, Anikó and Varga, Csaba and Kupai, Krisztina (2021) Effects of aging on proteasomal-ubiquitin system, oxidative stress balance and calcium homeostasis in middle-aged female rat colon. Physiology International, 108 (1). pp. 27-42. ISSN 2498-602X

Szabó, Írisz and Varga, Viktória É. and Dvorácskó, Szabolcs and Farkas, Elek Attila and Körmöczi, Tímea and Berkecz, Róbert and Kecskés, Szilvia and Menyhárt, Ákos and Frank, Rita and Frecska, Ede and Tömböly, Csaba and Krizbai, István Adorján and Bari, Ferenc and Farkas, Eszter (2021) N,N-Dimethyltryptamine attenuates spreading depolarization and restrains neurodegeneration by sigma-1 receptor activation in the ischemic rat brain. NEUROPHARMACOLOGY, 192. ISSN 0028-3908

Dvorácskó, Szabolcs and Lázár, László and Fülöp, Ferenc and Palkó, Márta and Zalán, Zita and Penke, Botond and Fülöp, Lívia and Tömböly, Csaba and Bogár, Ferenc (2021) Novel High Affinity Sigma-1 Receptor Ligands from Minimal Ensemble Docking-Based Virtual Screening. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 22 (15). pp. 1-17. ISSN 1661-6596 (print); 1422-0067 (online)

Zádor, Ferenc and Joca, Sâmia and Nagy-Grócz, Gábor and Dvorácskó, Szabolcs and Szűcs, Edina and Tömböly, Csaba and Benyhe, Sándor and Vécsei, László (2021) Pro-Inflammatory Cytokines: Potential Links between the Endocannabinoid System and the Kynurenine Pathway in Depression. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 22 (11). ISSN 1661-6596

Almási, Nikoletta and Török, Szilvia and Dvorácskó, Szabolcs and Tömböly, Csaba and Csonka, Ákos and Baráth, Zoltán Lajos and Murlasits, Zsolt and Valkusz, Zsuzsanna and Pósa, Anikó and Varga, Csaba and Kupai, Krisztina (2020) Lessons on the Sigma-1 Receptor in TNBS-Induced Rat Colitis. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 21 (11). ISSN 1661-6596

Zádor, Ferenc and Nagy-Grócz, Gábor and Dvorácskó, Szabolcs and Bohár, Zsuzsanna and Cseh, Edina Katalin and Zádori, Dénes and Párdutz, Árpád and Szűcs, Edina and Tömböly, Csaba and Borsodi, Anna and Benyhe, Sándor and Vécsei, László (2020) Long-term systemic administration of kynurenic acid brain region specifically elevates the abundance of functional CB1 receptors in rats. NEUROCHEMISTRY INTERNATIONAL, 138. ISSN 0197-0186

Herman, Bianka Edina and Gardi, János and Julesz, János and Tömböly, Csaba and Szánti-Pintér, Eszter and Fehér, Klaudia and Skoda-Földes, Rita and Szécsi, Mihály (2020) Steroidal Ferrocenes as Potential Enzyme Inhibitors of the Estrogen Biosynthesis. BIOLOGIA FUTURA, 71 (3). pp. 249-264. ISSN 2676-8615 (print); 2676-8607 (online)

Szűcs, Edina and Marton, János and Szabó, Zoltán and Hosztafi, Sándor and Kékesi, Gabriella and Bánki, László and Horváth, Gyöngyi and Szabó, Pál Tamás and Tömböly, Csaba and Benyhe, Sándor and Ötvös, Ferenc and Tuboly, Gábor and Varga, Zsuzsanna Katalin (2020) Synthesis, biochemical, pharmacological characterization and in silico profile modelling of highly potent opioid orvinol and thevinol derivatives. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 191. ISSN 0223-5234

Dimmito, Marilisa P. and Stefanucci, Azzurra and Pieretti, Stefano and Minosi, Paola and Dvorácskó, Szabolcs and Tömböly, Csaba and Zengin, Gokhan and Mollica, Adriano (2019) Discovery of Orexant and Anorexant Agents with Indazole Scaffold Endowed with Peripheral Antiedema Activity. BIOMOLECULES, 9 (9). ISSN 2218-273X

Zádor, Ferenc and Nagy-Grócz, Gábor and Kékesi, Gabriella and Dvorácskó, Szabolcs and Szűcs, Edina and Tömböly, Csaba and Horváth, Gyöngyi and Benyhe, Sándor and Vécsei, László (2019) Kynurenines and the Endocannabinoid System in Schizophrenia: Common Points and Potential Interactions. MOLECULES, 24 (20). pp. 1-36. ISSN 1420-3049

Dvorácskó, Szabolcs and Keresztes, Attila and Mollica, Adriano and Stefanucci, Azzurra and Macedonio, Giorgia and Zádor, Ferenc and Walter, Fruzsina R. and Deli, Mária A. and Kékesi, Gabriella and Bánki, László and Tuboly, Gábor and Horváth, Gyöngyi and Tömböly, Csaba (2019) Preparation of bivalent agonists for targeting the mu opioid and cannabinoid receptors. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 178. pp. 571-588. ISSN 0223-5234

Stefanucci, Azzurra and Novellino, Ettore and Macedonio, Giorgia and Dimmito, Marilisa Pia and Mirzaie, Sako and Cardoso, Fernanda Caldas and Lewis, Richard and Zádor, Ferenc and Erdei, Anna and Dvorácskó, Szabolcs and Tömböly, Csaba and Benyhe, Sándor and Pieretti, Stefano and Minosi, Paola and Mollica, Adriano (2018) Design, synthesis and biological profile of mixed opioid agonist/N-VGCC blocker peptides. NEW JOURNAL OF CHEMISTRY, 42 (8). pp. 5656-5659. ISSN 1144-0546

De Prins, A. and Martin, C. B. and Van Wanseele, Y and Skov, L. J. and Tömböly, Csaba (2018) Development of potent and proteolytically stable human neuromedin U receptor agonists. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 144. pp. 887-897. ISSN 0223-5234

Leone, Sheila and Ferrante, Claudio and Recinella, Lucia and Chiavaroli, Annalisa and Mollica, Adriano and Tömböly, Csaba and Stefanucci, Azzurra and Dimmito, Marilisa Pia and Dvorácskó, Szabolcs and Verratti, Vittore and De Petrocellis, Luciano and Orlando, Giustino and Brunetti, Luigi (2018) Effects of RVD-hemopressin (α) on feeding and body weight after standard or cafeteria diet in rats. NEUROPEPTIDES, 72. pp. 38-46. ISSN 0143-4179

Corbani, M. and Marir, R. and Truebai, M. and Chafai, M. and Vincent, A. and Tömböly, Csaba (2018) Neuroanatomical distribution and function of the vasopressin V-1B receptor in the rat brain deciphered using specific fluorescent ligands. GENERAL AND COMPARATIVE ENDOCRINOLOGY, 258. pp. 15-32. ISSN 0016-6480

Stefanucci, Azzurra and Macedonio, Giorgia and Dvorácskó, Szabolcs and Tömböly, Csaba and Mollica, Adriano (2018) Novel Fubinaca/Rimonabant hybrids as endocannabinoid system modulators. AMINO ACIDS, 50 (11). pp. 1595-1605. ISSN 0939-4451

De Prins, An and Martin, Charlotte and Van Wanseele, Yannick and Tömböly, Csaba and Tourwé, Dirk and Caveliers, Vicky and Holst, Birgitte and Van Eeckhaut, Ann and Rosenkilde, Mette Marie and Smolders, Ilse and Ballet, Steven (2018) Synthesis and in Vitro Evaluation of Stabilized and Selective Neuromedin U-1 Receptor Agonists. ACS MEDICINAL CHEMISTRY LETTERS, 9 (5). pp. 496-501. ISSN 1948-5875

Bacsa, Ildikó and Herman, Bianka Edina and Jójárt, Rebeka and Herman, Kevin Stefán and Wölfling, János and Schneider, Gyula and Varga, Mónika and Tömböly, Csaba and Szécsi, Mihály and Mernyák, Erzsébet (2018) Synthesis and structure–activity relationships of 2- and/or 4-halogenated 13β- and 13α-estrone derivatives as enzyme inhibitors of estrogen biosynthesis. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 33 (1). pp. 1271-1282. ISSN 1475-6366 (print); 1475-6374 (online)

Adamska-Bartlomiejczyk, Anna and Janecka, Anna and Szabó, Márton Richárd and Tömböly, Csaba and Borics, Attila (2017) Cyclic mu-opioid receptor ligands containing multiple N-methylated amino acid residues. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 27 (8). pp. 1644-1648. ISSN 0960-894X

Mollica, A. and Pelliccia, S. and Famiglini, V. and Stefanucci, A. and Macedonio, G. and Benyhe, Sándor and Zádor, Ferenc and Erdei, Anna and Szűcs, Edina and Samavati, Reza and Dvorácskó, Szabolcs and Tömböly, Csaba (2017) Exploring the first Rimonabant analog-opioid peptide hybrid compound, as bivalent ligand for CB1 and opioid receptors. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 32 (1). pp. 444-451. ISSN 1475-6366

Adamska-Bartlomiejczyk, Anna and Borics, Attila and Tömböly, Csaba and Dvorácskó, Szabolcs and Lisowski, Marek (2017) Synthesis, receptor binding studies, optical spectroscopic and in silico structural characterization of morphiceptin analogs with cis-4-amino-L-proline residues. JOURNAL OF PEPTIDE SCIENCE, 23 (12). pp. 864-870. ISSN 1075-2617

Szűcs, Edina and Dvorácskó, Szabolcs and Tömböly, Csaba and Büki, Alexandra and Kékesi, Gabriella and Horváth, Gyöngyi and Benyhe, Sándor (2016) Decreased CB receptor binding and cannabinoid signaling in three brain regions of a rat model of schizophrenia. NEUROSCIENCE LETTERS, 633. pp. 87-93. ISSN 0304-3940

Monti, L. and Stefanucci, A. and Pieretti, S. and Marzoli, F. and Fidanza, L. and Benyhe, Sándor and Zádor, Ferenc and Szűcs, Edina and Ötvös, Ferenc and Erdei, Anna and Samavati, Reza and Dvorácskó, Szabolcs and Tömböly, Csaba (2016) Evaluation of the analgesic effect of 4-anilidopiperidine scaffold containing ureas and carbamates. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 31 (6). pp. 1638-1647. ISSN 1475-6366

Dvorácskó, Szabolcs and Tömböly, Csaba and Berkecz, Róbert and Keresztes, Attila (2016) Investigation of receptor binding and functional characteristics of hemopressin(1-7). NEUROPEPTIDES, 58. pp. 15-22. ISSN 0143-4179

Piekielna, Justyna and De Marco, Rossella and Gentilucci, Luca and Cerlesi, Maria Camilla and Calo', G. and Tömböly, Csaba (2016) Redoubling the Ring Size of an Endomorphin-2 Analog Transforms a Centrally Acting Mu-Opioid Receptor Agonist into a Pure Peripheral Analgesic. BIOPOLYMERS, 106 (3). pp. 309-317. ISSN 0006-3525

Schäfer, Balázs and Orbán, Erika and Fiser, Gabriella and Marton, Annamária and Vizler, Csaba and Tömböly, Csaba (2016) Semisynthesis of membrane-anchored cholesteryl lipoproteins on live cell surface by azide–alkyne click reaction. TETRAHEDRON LETTERS, 57 (8). pp. 868-873. ISSN 0040-4039

Perlikowska, Renata and Piekielna, Justyna and Gentilucci, Luca and De Marco, Rossella and Cerlesi, Maria Camilla and Tömböly, Csaba (2016) Synthesis of mixed MOR/KOR efficacy cyclic opioid peptide analogs with antinociceptive activity after systemic administration. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 109. pp. 276-286. ISSN 0223-5234

Szlávicz, Eszter and Perera, Pannilage Shiromi and Tömböly, Csaba and Helyes, Zsuzsanna and Zádor, Ferenc and Benyhe, Sándor and Borsodi, Anna and Bojnik, Engin (2015) Further Characterization of Hemopressin Peptide Fragments in the Opioid and Cannabinoid Systems. ANESTHESIA AND ANALGESIA, 121 (6). pp. 1488-1494. ISSN 0003-2999

Piekielna, J. and Kluczyk, A. and Gentilucci, L. and Cerlesi, M.C. and Calo', G. and Tömböly, Csaba (2015) Ring size in cyclic endomorphin-2 analogs modulates receptor binding affinity and selectivity. ORGANIC & BIOMOLECULAR CHEMISTRY, 13 (21). pp. 6039-6046. ISSN 1477-0520

Piekielna, Justyna and Perlikowska, Renata and do-Rego, Jean-Claude and do-Rego, Jean-Luc and Cerlesi, Maria Camilla and Tömböly, Csaba (2015) Synthesis of Mixed Opioid Affinity Cyclic Endomorphin-2 Analogues with Fluorinated Phenylalanines. ACS MEDICINAL CHEMISTRY LETTERS, 6 (5). pp. 579-583. ISSN 1948-5875

Keresztes, Attila and Borics, Attila and Tömböly, Csaba (2015) Therapeutic and diagnostic radiopharmaceuticals. In: Selected Topics from Contemporary Experimental Biology. MTA Szegedi Biológiai Központ, Szeged, pp. 225-247.

Schäfer, Balázs and Orban, E. and Kele, Zoltán and Tömböly, Csaba (2015) Tritium labelling of a cholesterol amphiphile designed for cell membrane anchoring of proteins. JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS, 58 (1). pp. 7-13. ISSN 0362-4803

Piekielna, Justyna and Gentilucci, Luca and De Marco, Rossella and Perlikowska, Renata and Adamska, Anna and Tömböly, Csaba (2014) Cyclic side-chain-linked opioid analogs utilizing cis- and trans-4-aminocyclohexyl-D-alanine. BIOORGANIC AND MEDICINAL CHEMISTRY, 22 (23). pp. 6545-6551. ISSN 0968-0896

Ballet, Steven and Betti, Cecilia and Novoa, Alexandre and Tömböly, Csaba and Uhd, Nielsen (2014) In Vitro Membrane Permeation Studies and in Vivo Antinociception of Glycosylated Dmt1-DALDA Analogues. ACS MEDICINAL CHEMISTRY LETTERS, 5 (4). pp. 352-357. ISSN 1948-5875

Perlikowska, R. and Malfacini, D. and Cerlesi, M. C. and Calo', G. and Piekielna, J. and Tömböly, Csaba (2014) Pharmacological characterization of endomorphin-2-based cyclic pentapeptides with methylated phenylalanine residues. PEPTIDES, 55C. pp. 145-150. ISSN 0196-9781

Schäfer, Balázs and Orbán, Erika and Borics, Attila and Huszár, Krisztina and Nyeste, Antal and Welker, Ervin and Tömböly, Csaba (2013) Preparation of semisynthetic lipoproteins with fluorescent cholesterol anchor and their introduction to the cell membrane with minimal disruption of the membrane. Bioconjugate Chemistry, 24 (10). pp. 1684-1697. ISSN 1043-1802

Tömböly, Csaba (2009) Fehérjék előállítása kémiai módszerekkel szerkezeti és funkcionális vizsgálatok céljára = Total synthesis of proteins for structural and functional studies. Project Report. OTKA.

Tóth, Géza and Farkas, Judit and Hunyadi-Gulyás, Éva Csilla and Ötvös, Ferenc and Péter, Antal and Szemenyei, Erzsébet and Tömböly, Csaba (2008) Neuropeptidek radioaktív jelölése = Radioactive labelling of neuropeptides. Project Report. OTKA.

This list was generated on Fri Mar 29 12:08:20 2024 CET.