Items where Author is "Wölfling, János"

Article

Nagymihály, Zoltán and Wölfling, János and Schneider, Gyula and Kollár, László (2020) Synthesis of 2-Methylresorcinol-Based Deepened Cavitands with Chiral Inlet Bearing Steroidal Moieties on the Upper Rim. ChemistrySelect. pp. 6933-6938. ISSN 2365-6549

Herman, Bianka Edina and Kiss, Anita and Wölfling, János and Mernyák, Erzsébet and Szécsi, Mihály and Schneider, Gyula (2019) Synthesis of substituted 15β-alkoxy estrone derivatives and their cofactor-dependent inhibitory effect on 17β-HSD1. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 34 (1). pp. 1271-1286. ISSN 1475-6366

Angyal, Anikó and Demjén, András and Harmat, Veronika and Wölfling, János and Puskás, László G. and Kanizsai, Iván (2019) 1,3-Dipolar Cycloaddition of Isatin-Derived Azomethine Ylides with 2H‐Azirines: Stereoselective Synthesis of 1,3- Diazaspiro[bicyclo[3.1.0]hexane]oxindoles. JOURNAL OF ORGANIC CHEMISTRY, 84 (7). pp. 4273-4281. ISSN 0022-3263

Demjén, András and Alföldi, Róbert and Angyal, Anikó and Gyuris, Márió and Hackler, László, Jr. and Szebeni, Gábor J. and Wölfling, János and Kanizsai, Iván and Puskás, László G. (2018) Synthesis, cytotoxic characterization, and SAR study of imidazo[1,2-b]pyrazole-7-carboxamides. ARCHIV DER PHARMAZIE. pp. 1-21. ISSN 0365-6233

Bacsa, Ildikó and Szemerédi, Dávid and Wölfling, János and Schneider, Gyula and Fekete, Lilla and Mernyák, Erzsébet (2018) The first Pd-catalyzed Buchwald–Hartwig aminations at C-2 or C-4 in the estrone series. BEILSTEIN JOURNAL OF ORGANIC CHEMISTRY. ISSN 1860-5397

Bacsa, Ildikó and Herman, Bianka Edina and Jójárt, Rebeka and Herman, Kevin Stefán and Wölfling, János and Schneider, Gyula and Varga, Mónika and Tömböly, Csaba and Szécsi, Mihály and Mernyák, Erzsébet (2018) Synthesis and structure–activity relationships of 2- and/or 4-halogenated 13β- and 13α-estrone derivatives as enzyme inhibitors of estrogen biosynthesis. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 33 (1). pp. 1271-1282. ISSN 1475-6366 (print); 1475-6374 (online)

Fröhlich, Tony and Kiss, Anita and Wölfling, János and Mernyák, Erzsébet and Kulmány, Ágnes E. and Minorics, Renáta and Zupkó, István and Schneider, Gyula (2018) Synthesis of Artemisinin-Estrogen Hybrids Highly Active against HCMV, P. falciparum, and Cervical and Breast Cancer. ACS MEDICINAL CHEMISTRY LETTERS, 9 (11). pp. 1-6. ISSN 1948-5875

Demjén, András and Alföldi, Róbert and Angyal, Anikó and Gyuris, Márió and Hackler, László and Szebeni, Gábor J. and Wölfling, János and Puskás, László G. and Kanizsai, Iván (2018) Synthesis, cytotoxic characterization, and SAR study of imidazo[1,2-b]pyrazole-7-carboxamides. ARCHIV DER PHARMAZIE, 351 (7). pp. 1-21. ISSN 0365-6233

Bózsity, Noémi and Minorics, Renáta and Szabó, Johanna and Mernyák, Erzsébet and Schneider, Gyula and Wölfling, János and Ocsovszki, Imre and Zupkó, István (2017) Mechanism of antiproliferative action of a new D-secoestrone-triazole derivative in cervical cancer cells and its effect on cancer cell motility. JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 165. pp. 247-257. ISSN 0960-0760

Bacsa, Ildikó and Jójárt, Rebeka and Wölfling, János and Schneider, Gyula and Herman, Bianka Edina and Szécsi, Mihály and Mernyák, Erzsébet (2017) Synthesis of novel 13 α-estrone derivatives by Sonogashira coupling as potential 17 β-HSD1 inhibitors. BEILSTEIN JOURNAL OF ORGANIC CHEMISTRY, 13. pp. 1303-1309. ISSN 1860-5397

Bózsity, Noémi and Minorics, Renáta and Szabó, Johanna and Mernyák, Erzsébet and Schneider, Gyula and Wölfling, János and Wang, Hui-Chun and Wu, Chin-Chung and Ocsovszki, Imre and Zupkó, István (2016) Mechanism of antiproliferative action of a new D-secoestrone-triazole derivative in cervical cancer cells and its effect on cancer cell motility. JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY. ISSN 0960-0760 (In Press)

Baji, Ádám and Gyovai, András and Wölfling, János and Minorics, Renáta and Ocsovszki, Imre and Zupkó, István and Frank, Éva (2016) Microwave-assisted one-pot synthesis of steroid– quinoline hybrids and an evaluation of their antiproliferative activities on gynecological cancer cell lines. RSC Advances, 6. pp. 27501-27516. ISSN 2046-2069

Baji, Ádám and Gyovai, András and Wölfling, János and Minorics, Renáta and Ocsovszki, Imre and Zupkó, István and Frank, Éva (2016) Microwave-assisted one-pot synthesis of steroid–quinoline hybrids and an evaluation of their antiproliferative activities on gynecological cancer cell lines. RSC ADVANCES. pp. 1-50. ISSN 2046-2069

Schneider, Gyula and Kiss, Anita and Mernyák, Erzsébet and Benke, Zsanett and Wölfling, János and Frank, Éva and Bózsity, Noémi and Gyovai, András and Minorics, Renáta and Zupkó, István (2016) Stereocontrolled synthesis of the four 16-hydroxymethyl-19- nortestosterone isomers and their antiproliferative activities. STEROIDS, 105. pp. 113-120. ISSN 0039-128X

Schneider, Gyula and Kiss, Anita and Mernyák, Erzsébet and Benke, Zsanett and Wölfling, János and Frank, Éva and Bózsity, Noémi and Gyovai, András and Minorics, Renáta and Zupkó, István (2016) Stereocontrolled synthesis of the four 16-hydroxymethyl-19-nortestosterone isomers and their antiproliferative activities. STEROIDS, 105. pp. 113-120. ISSN 0039-128X

Szabó, Johanna and Pataki, Zoltán and Wölfling, János and Schneider, Gyula and Bózsity, Noémi and Minorics, Renáta and Zupkó, István and Mernyák, Erzsébet (2016) Synthesis and biological evaluation of 13a-estrone derivatives as potential antiproliferative agents. STEROIDS, 113. pp. 14-21. ISSN 0039-128X

Szabó, Johanna and Pataki, Zoltán and Wölfling, János and Schneider, Gyula and Bózsity, Noémi and Minorics, Renáta and Zupkó, István and Mernyák, Erzsébet (2016) Synthesis and biological evaluation of 13α-estrone derivatives as potential antiproliferative agents. STEROIDS, 113. pp. 14-21. ISSN 0039-128X

Szabó, Johanna and Jerkovics, Nóra and Schneider, Gyula and Wölfling, János and Bózsity, Noémi and Minorics, Renáta and Zupkó, István and Mernyák, Erzsébet (2016) Synthesis and in Vitro Antiproliferative Evaluation of C-13 Epimers of Triazolyl-D-Secoestrone Alcohols: The First Potent 13α-D-Secoestrone Derivative. MOLECULES, 21 (611). ISSN 1420-3049

Szabó, Johanna and Jerkovics, Nóra and Schneider, Gyula and Wölfling, János and Bózsity, Noémi and Minorics, Renáta and Zupkó, István and Mernyák, Erzsébet (2016) Synthesis and in Vitro Antiproliferative Evaluation of C-13 Epimers of Triazolyl-D-Secoestrone Alcohols: The First Potent 13α-D-Secoestrone Derivative. MOLECULES, 21 (5). pp. 1-13. ISSN 1420-3049

Molnár, Judit and Nagyné, Frank Éva and Minorics, Renáta and Kádár, Zalán and Ocsovszki, Imre and Wölfling, János and Zupkó, István (2015) A Click Approach to Novel D-Ring-Substituted 16α-Triazolylestrone Derivatives and Characterization of Their Antiproliferative Properties. PLOS ONE, 10 (2). e0118104. ISSN 1932-6203

Kovács, Dóra Irén and Wölfling, János and Szabó, N. and Szécsi, M. and Minorics, Renáta and Zupkó, István and Nagyné, Frank Éva (2015) Efficient access to novel androsteno-17-(1′,3′,4′)-oxadiazoles and 17<beta>-(1′,3′,4′)-thiadiazoles via N-substituted hydrazone and N,N′-disubstituted hydrazine intermediates, and their pharmacological evaluation in vitro. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 98. pp. 13-29. ISSN 0223-5234

Mótyán, Gergő and Zupkó, István and Minorics, Renáta and Schneider, Gyula and Wölfling, János and Frank, Éva (2015) Lewis acid-induced intramolecular access to novel steroidal ring D-condensed arylpyrazolines exerting in vitro cell-growth-inhibitory effects. MOLECULAR DIVERSITY .

Szabó, Nikoletta and Iványi, Zoltán and Szécsi, Mihály and Julesz, János and Mernyák, Erzsébet and Huber, Judit and Wölfling, János and Minorics, Renáta and Zupkó, István and Schneider, Gyula (2015) Synthesis of methoxycarbonylpyrazolylandrostene derivatives, and their potential inhibitory effect on androgen biosynthesis and cell proliferation. STEROIDS, 98. pp. 143-152. ISSN 0039-128X

Schneider, Gyula and Görbe, Tamás and Mernyák, Erzsébet and Wölfling, János and Holczbauer, Tamás and Minorics, Renáta and Zupkó, István (2015) Synthesis of novel 17-(5’-iodo)triazolyl-3-methoxyestrane epimers via Cu(I)-catalyzed azide-alkyne cycloadditon, and an evaluation of their cytotoxic activity in vitro. STEROIDS, 98. pp. 153-165. ISSN 0039-128X

Mernyák, Erzsébet and Kovács, Ida and Minorics, Renáta and Sere, Péter and Czégány, Dóra and Wölfling, János and Schneider, Gyula and Újfaludi, Zsuzsanna and Boros, Imre Miklós and Zupkó, István (2015) Synthesis of trans-16-triazolyl-13α-methyl-17-estradiol diastereomers and the effects of structural modifications on their in vitro antiproliferative activities. JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 150. pp. 123-134. ISSN 0960-0760

Minorics, Renáta and Bózsity, Noémi and Molnár, Judit and Wölfling, János and Mernyák, Erzsébet and Zupkó, István (2015) A molecular understanding of d-homoestrone-induced G2/M cell cycle arrest in HeLa human cervical carcinoma cells. JOURNAL OF CELLULAR AND MOLECULAR MEDICINE, in pre. 10.1111/jcmm.12587. ISSN 1582-1838

Iványi, Zoltán and Görbe, Tamás and Szabó, Nikoletta and Kiss, Anita and Wölfling, János and Schneider, Gyula (2014) 17ß-Pirazolil- és -pirazolinil-szteroidok szintézise. MAGYAR KÉMIAI FOLYÓIRAT - KÉMIAI KÖZLEMÉNYEK, 120 (2-3). pp. 116-121. ISSN 1418-9933

Madácsi, Ramóna and Gyuris, Márió and Kanizsai, Iván and Sipos, Péter and Wölfling, János (2014) 4-Amino-5,6,7-trifluor-ftálimidek előállítása, in vitro és in vivo biológiai vizsgálata. MAGYAR KÉMIAI FOLYÓIRAT - KÉMIAI KÖZLEMÉNYEK, 120 (2-3). pp. 95-101. ISSN 1418-9933

Wölfling, János (2014) A Szegedi Tudományegyetem Kémia Doktori Iskolája. MAGYAR KÉMIAI FOLYÓIRAT - KÉMIAI KÖZLEMÉNYEK, 120 (2-3). p. 44. ISSN 1418-9933

Juhász-Vedres, Gabriella and Rózsa, Éva and Rákos, Gabriella and Dobszay B., Gábor and Kis, Zsolt and Wölfling, János and Toldi, József and Párducz, Árpád and Farkas, Tamás (2006) Dehydroepiandrosterone sulfate (DHEAS) is neuroprotective when administered either before or after injury in a focal cortical cold lesion model. Endocrinology, 147 (2). pp. 683-686. ISSN 0013-7227 (print), 1945-7170 (online)

Monograph

Schneider, Gyula and Nagyné dr. Frank, Éva and Wölfling, János (2011) Szteránvázas vegyületek kutatása = Research of steroids. Project Report. OTKA.

Wölfling, János and Julesz, János and Mernyák, Erzsébet and Nagyné dr. Frank, Éva and Schneider, Gyula and Szájli, Ágota and Szécsi, Mihály and Tóth, István (2009) Antiandrogén kardenolid analógok szintézise és biológiai hatásvizsgálata = Synthesis and biological effect investigations of antiandrogen cardenolide analogues. Project Report. OTKA.

Schneider, Gyula and Magyar, Angéla Andrea and Mernyák, Erzsébet and Nagyné dr. Frank, Éva and Wölfling, János (2007) Szteránvázas vegyületek szintézise = Synthesis of Steroid Compounds. Project Report. OTKA.

Conference or Workshop Item

Farkas, Tamás and Juhász-Vedres, Gabriella and Rózsa, Éva and Rákos, Gabriella and Kis, Zsolt and Wölfling, János and Toldi, József (2007) Dehydroepiandrosterone sulfate is neuroprotective in a focal cortical cold lesion model. In: Göttingen Meeting of the German Neuroscience Society 2007: 31st Göttingen Neurobiology Conference, 2007.03.29-2007.04.01, Göttingen, Németország.