Items where Author is "Somsák, László"

József, János and Somsák, László and Juhász, János (2023) Exo-glikál származékok átalakításainak a vizsgálata: tioladdíciós és cikloaddíciós reakciók. MAGYAR KÉMIAI FOLYÓIRAT - KÉMIAI KÖZLEMÉNYEK (1997-), 129 (3-4). pp. 147-154. ISSN 1418-9933

Kiss, Mariann and Timári, István and Barna, Teréz and Mészáros, Zuzana and Slámová, Kristýna and Somsák, László (2022) 2-Acetamido-2-deoxy-d-glucono-1,5-lactone Sulfonylhydrazones: Synthesis and Evaluation as Inhibitors of Human OGA and HexB Enzymes. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 23 (3). pp. 1-18. ISSN 1661-6596

Kiss, Mariann and Szabó, Erna and Bocska, Boglárka and Sinh, Luu Thanh and Fernandes, Conceicao Piedade and Timári, István and Somsák, László and Barna, Teréz (2021) Nanomolar inhibition of human OGA by 2-acetamido-2-deoxy-d-glucono-1,5-lactone semicarbazone derivatives. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 223. No.-113649. ISSN 0223-5234

Csávás, Magdolna and Eszenyi, Dániel and Mező, Erika and Lázár, László and Debreczeni, Nóra and Tóth, Marietta and Somsák, László and Borbás, Anikó (2020) Stereoselective Synthesis of Carbon-Sulfur-Bridged Glycomimetics by Photoinitiated Thiol-Ene Coupling Reactions. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 21. pp. 573-600. ISSN 1422-0067

Lázár, László and Juhász, László and Batta, Gyula and Borbás, Anikó and Somsák, László (2017) Unprecedented b-manno type thiodisaccharides with a C-glycosylic function by photoinitiated hydrothiolation of 1-C-substituted glycals. New Journal of Chemistry, 41 (3). pp. 1284-1292. ISSN 1144-0546, ESSN: 1369-9261

Nagy, Lilla Nikoletta and Márton, Judit and Vida, András and Kis, G. and Bokor, Éva and Kun, Sándor and Docsa, Tibor and Gergely, Pál and Pacher, Pál and Somsák, László and Bay, Péter (2017) Glycogen phosphorylase inhibition improves β-cell function. BRITISH JOURNAL OF PHARMACOLOGY. pp. 1-19. ISSN 0007-1188

Nagy, Veronika and Czifrák, Katalin and Apelt, Olena and Juhász, László and Somsák, László (2017) Preparation of glycosyl bromides of α-D-gluco-hept-2-ulopyranosonic acid derivatives. In: Carbohydrate Chemistry: Proven Synthetic Methods. CRC, pp. 69-75. ISBN 9781498726917 (In Press)

Agócs, Attila and Bokor, Éva and Takátsy, Anikó and Lóránd, Tamás and Deli, József and Somsák, László and Nagy, Veronika (2017) Synthesis of carotenoid-monosaccharide conjugates via azide–alkyne click-reaction. TETRAHEDRON, 73. pp. 519-526. ISSN 0040-4020

Lázár, László and József, János and Csávás, Magdolna and Tóth, Marietta and Juhász, László and Borbás, Anikó and Somsák, László (2015) SYNTHESIS OF CARBON-SULFUR-BRIDGED GLYCOMIMETICS BY THIOL-ENE COUPLING REACTIONS. In: Debrecen Colloquium on Carbohydrates 2015, András Lipták Memorial Conference, 2015. November 6-8., Debrecen.

Bokor, Éva and Szennyes, Eszter and Csupász, Tibor and Tóth, Nóra and Docsa, Tibor and Gergely, Pál and Somsák, László (2015) C-(2-Deoxy-D-arabino-hex-1-enopyranosyl)-oxadiazoles: synthesis of possible isomers and their evaluation as glycogen phosphorylase inhibitors. Carbohydrate Research, 412. pp. 71-79. ISSN 0008-6215

Misra, A. K. and Bokor, Éva and Kun, Sándor and Bolyog-Nagy, Evelin and Kathó, Ágnes and Joó, Ferenc and Somsák, László (2015) Chemoselective hydration of glycosyl cyanides to C-glycosyl formamides using ruthenium complexes in aqueous media. TETRAHEDRON LETTERS, 56 (44). pp. 5995-5998. ISSN 0040-4039

Begum, J. and Varga, G. and Docsa, Tibor and Gergely, Pál and Hayes, J. M. and Juhász, László and Somsák, László (2015) Computationally motivated synthesis and enzyme kinetic evaluation of N-(β-D-glucopyranosyl)-1,2,4-triazolecarboxamides as glycogen phosphorylase inhibitors. MEDCHEMCOMM, 6. pp. 80-89. ISSN 2040-2503

Somsák, László (2015) Előszó: Ezerarcú szénhidrátok. MAGYAR KÉMIAI FOLYÓIRAT - KÉMIAI KÖZLEMÉNYEK, 121 (1). p. 3. ISSN 1418-9933

Somsák, László and Pintér, István (2015) Szénhidrátok mindenütt. MAGYAR KÉMIAI FOLYÓIRAT - KÉMIAI KÖZLEMÉNYEK, 121 (1). pp. 27-33. ISSN 1418-9933

Lázár, László and Csávás, Magdolna and Tóth, Marietta and Somsák, László and Borbás, Anikó (2015) Thio-click approach to the synthesis of stable glycomimetics. Chemical Papers, 69 (6). pp. 889-895. ISSN 0366-6352, ESSN: 1336-9075

Czifrák, Katalin and Páhi, A. and Deák, Sz. and Kiss, Attila and E Kövér, Katalin and Docsa, Tibor and Gergely, Pál and Somsák, László (2014) Glucopyranosylidene-spiro-iminothiazolidinone, a new bicyclic ring system: synthesis, derivatization, and evaluation for inhibition of glycogen phosphorylase by enzyme kinetic and crystallographic methods. BIOORGANIC & MEDICINAL CHEMISTRY, 22. pp. 4028-4041. ISSN 0968-0896

Kun, Sándor and Bokor, Éva and Varga, G. and Szőcs, B. and Páhi, A. and Vágvölgyiné Tóth, Marietta and Juhász, László and Docsa, Tibor and Gergely, Pál and Somsák, László (2014) New synthesis of 3-(beta-D-glucopyranosyl)-5-substituted-1,2,4-triazoles, nanomolar inhibitors of glycogen phosphorylase. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 76. pp. 567-579. ISSN 0223-5234

Juhász, László and Varga, G. and Sztankovics, A. and Béke, F. and Docsa, Tibor and Kiss, Attila and Gergely, Pál and Somsák, László (2014) Structure-activity relationships of glycogen phosphorylase inhibitor FR258900 and its analogues: a combined synthetic, enzyme kinetics, and computational study. CHEMPLUSCHEM, 79 (11). pp. 1558-1568. ISSN 2192-6506

Somsák, László and Bokor, Éva and Czibere, B. and Czifrák, Katalin and Koppány, Cs. and Kun, Sándor and Vágvölgyiné Tóth, Marietta and Docsa, Tibor and Gergely, Pál (2014) Synthesis of C-xylopyranosyl- and xylopyranosylidene-spiro-heterocycles as potential inhibitors of glycogen phosphorylase. Carbohydrate Research, 399. pp. 38-48. ISSN 0008-6215

Varga, Gergely and Docsa, Tibor and Gergely, Pál and Juhász, László and Somsák, László (2013) Synthesis of tartaric acid analogues of FR258900 and their evaluation as glycogen phosphorylase inhibitors. Bioorganic & medicinal chemistry letters, 23 (6). pp. 1789-92. ISSN 1464-3405

Bokor, Éva and Docsa, Tibor and Gergely, Pál and Somsák, László (2013) C-Glucopyranosyl-1,2,4-triazoles As New Potent Inhibitors of Glycogen Phosphorylase. ACS MEDICINAL CHEMISTRY LETTERS, 4 (7). pp. 612-615. ISSN 1948-5875

Nagy, Lilla Nikoletta and Docsa, Tibor and Brunyánszki, Attila and Szántó, Magdolna and Hegedűs, Csaba and Márton, Judit and Virág, László and Somsák, László and Gergely, Pál and Bay, Péter (2013) Glycogen phosphorylase inhibitor N-(3,5-dimethyl-benzoyl)-N'-(β-Dglucopyranosyl) urea improves glucose tolerance under normoglycemic and diabetic conditions and rearranges hepatic metabolism. PLOS ONE, 8 (7). e69420. ISSN 1932-6203

Farkas, Etelka and Szabó, Orsolya and Tircsó, Gyula and Somsák, László (2013) Relaxometric determination of binding between Mn(II)–UDP and Mn(II)–UDP-glucose in aqueous solution. Carbohydrate Research, 368. pp. 68-72. ISSN 0008-6215

Tóth, Marietta and Szőcs, Béla and Kaszás, Tímea and Docsa, Tibor and Gergely, Pál and Somsák, László (2013) Synthesis of 2-(β-D-glucopyranosylamino)-5-substituted-1,3,4-oxadiazoles for inhibition of glycogen phosphorylase. CARBOHYDRATE RESEARCH, 381. pp. 196-204. ISSN 0008-6215

Szőcs, Béla and Tóth, Marietta and Docsa, Tibor and Gergely, Pál and Somsák, László (2013) Synthesis of 2-(β-d-glucopyranosyl)-5-(substituted-amino)-1,3,4-oxa- and -thiadiazoles for the inhibition of glycogen phosphorylase. CARBOHYDRATE RESEARCH, 381. pp. 187-195. ISSN 0008-6215

Bokor, Éva and Szilágyi, Enikő and Docsa, Tibor and Gergely, Pál and Somsák, László (2013) Synthesis of substituted 2-(β-d-glucopyranosyl)-benzimidazoles and their evaluation as inhibitors of glycogen phosphorylase. Carbohydrate Research, 381. pp. 179-186. ISSN 0008-6215

Varga, G. and Docsa, Tibor and Gergely, Pál and Juhász, László and Somsák, László (2013) Synthesis of tartaric acid analogues of FR258900 and their evaluation as glycogen phosphorylase inhibitors. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 23. pp. 1789-1792. ISSN 0960-894X

Polyák, M. and Varga, G. and Szilágyi, Bence and Juhász, László and Docsa, Tibor and Gergely, Pál and Somsák, László (2013) Synthesis, enzyme kinetics and computational evaluation of N-(beta-D-glucopyranosyl) oxadiazolecarboxamides as glycogen phosphorylase inhibitors. BIOORGANIC & MEDICINAL CHEMISTRY, 21. pp. 5738-5747. ISSN 0968-0896

Antus, Sándor and Czifrák, Katalin and Jakab, Zsolt and Kenéz, Ágnes and Kiss, Attila and Kónya, Krisztina Emília and Patonay, Tamás and Sipos, Attila and Somsák, László and Szabó, Ildikó Erzsébet and Varga, Gergely Tibor and Vasas, Attila (2010) Potenciálisan biológiailag aktív természetes anyagok és rokon vegyületeik kémiájának tanulmányozása = Study of the Chemistry of Natural Products and Related Compounds of Potential Biological Activity. Project Report. OTKA.

Somsák, László and Czifrák, Katalin and Györgydeák, Zoltán and Hadady, Zsuzsa and Nagy, Veronika and Vágvölgyiné dr.Tóth, Marietta (2008) Glikoenzim-inhibítorok előállítása = Synthesis of glycoenzyme inhibitors. Project Report. OTKA.

Micskei, Károly and Hajdu, Csongor and Somsák, László (2008) Szelektív szintézismódszerek kifejlesztése vizes közegben átmenetifém-komplexek jelenlétében = Development of selective synthetic methods in aqueous medium in the presence os transition metal complexes. Project Report. OTKA.

Somsák, László and Czifrák, Katalin and Györgydeák, Zoltán and Vágvölgyiné dr.Tóth, Marietta (2007) Glikozil-azidok szerepe az anomer szénatomhoz nitrogénen kötődő funkciós csoportok kialakításában = Role of glycosyl azides in the formation of N-bound functional groups at the anomeric centre. Project Report. OTKA.