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Items where Author is "Dvorácskó, Szabolcs"

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Herrerias, Alexa and Oliverio, Anna and Dvorácskó, Szabolcs and Thyagarajan, Arthi and Chedester, Lee and Liu, Jie and Cinar, Resat and Iyer, Malliga R. and Kunos, George and Godlewski, Grzegorz (2025) CB1 receptors on a subset of vagal afferent neurons modulate voluntary ethanol intake in mice. MOLECULAR PSYCHIATRY. ISSN 1359-4184

Bhattacharjee, Pinaki and Dvorácskó, Szabolcs and Pointeau, Oceane and Kundu, Biswajit and Rutland, Nicholas and Puhl, Henry and Liu, Jie and Godlewski, Grzegorz and Hassan, Sergio A. and Jourdan, Tony and Cinar, Resat and Iyer, Malliga R. (2025) Evaluation of tetrahydropyridazine-based peripherally restricted dual inhibitors of CB1R and inducible nitric oxide synthase (iNOS) for treating metabolic syndrome disorders. METABOLISM-CLINICAL AND EXPERIMENTAL, 170. No. -156291. ISSN 0026-0495

Sarkar, Arijit and Dvorácskó, Szabolcs and Lipinszki, Zoltán and Mitra, Argha and Harmati, Mária and Buzás, Krisztina and Borics, Attila (2025) Evidencing the role of a conserved polar signaling channel in the activation mechanism of the μ-opioid receptor. COMPUTATIONAL AND STRUCTURAL BIOTECHNOLOGY JOURNAL, 27. pp. 3216-3228. ISSN 2001-0370

Maccioni, Luca and Dvorácskó, Szabolcs and Godlewski, Grzegorz and Cinar, Resat and Iyer, Malliga R and Gao, Bin and Kunos, George (2025) Gut cannabinoid receptor 1 regulates alcohol binge-induced intestinal permeability. EGASTROENTEROLOGY, 3 (1). No. e100173. ISSN 2976-7296

Basu, Abhishek and Arif, Muhammad and Wolf, Kaelin M. and Behee, Madeline and Johnson, Natalie and Pommerolle, Lenny and Pineda, Ricardo H. and Sembrat, John and Zawatsky, Charles N. and Dvorácskó, Szabolcs and Coffey, Nathan J. and Park, Joshua K. and Karagoz, Seray B. and Godlewski, Grzegorz and Jourdan, Tony and Harvey-White, Judith and Königshoff, Melanie and Iyer, Malliga R. and Cinar, Resat (2025) Targeting cannabinoid receptor 1 for antagonism in pro-fibrotic alveolar macrophages mitigates pulmonary fibrosis. JCI INSIGHT, 10 (15). ISSN 2379-3708

Kecskés, Szilvia and Mészáros, Mária and Dvorácskó, Szabolcs and Szabó, Írisz and Porkoláb, Gergő and Barna, Lilla and Harazin, András and Szecskó, Anikó and Menyhárt, Ákos and Bari, Ferenc and Deli, Mária Anna and Penke, Botond and Farkas, Eszter and Veszelka, Szilvia (2025) The impact of the novel sigma1 receptor ligand (S)-L1 on brain endothelial cells and cerebrovascular reactivity challenged by ischemia. EUROPEAN JOURNAL OF PHARMACOLOGY, 1000. No.-177724. ISSN 0014-2999

Kumari, Punita and Dvorácskó, Szabolcs and Enos, Michael D. and Ramesh, Karthik and Lim, Darrix and Hassan, Sergio A. and Kunos, George and Cinar, Resat and Iyer, Malliga R. and Rosenbaum, Daniel M. (2024) Structural mechanism of CB1R binding to peripheral and biased inverse agonists. NATURE COMMUNICATIONS, 15 (1). No.-10694. ISSN 2041-1723

Dvorácskó, Szabolcs and Herrerias, A. and Oliverio, A. and Bhattacharjee, P. and Pommerolle, L. and Liu, Z. and Feng, D. and Lee, Y.-S. and Hassan, S.A. and Godlewski, G. and Cinar, R. and Iyer, M.R. (2023) Cannabinoformins: Designing Biguanide-Embedded, Orally Available, Peripherally Selective Cannabinoid-1 Receptor Antagonists for Metabolic Syndrome Disorders. JOURNAL OF MEDICINAL CHEMISTRY, 66 (17). pp. 11985-12004. ISSN 0022-2623

Dvorácskó, Szabolcs and Körmöczi, Tímea and Sija, Éva and Bende, Balázs and Weiczner, Roland and Varga, Tibor and Ilisz, István and Institóris, László and Kereszty, Éva M. and Tömböly, Csaba and Berkecz, Róbert (2023) Focusing on the 5F-MDMB-PICA, 4F-MDMB-BICA Synthetic Cannabinoids and Their Primary Metabolites in Analytical and Pharmacological Aspects. TOXICOLOGY AND APPLIED PHARMACOLOGY, 470. No.-116548. ISSN 0041-008X (print); 1096-0333 (online)

Dvorácskó, Szabolcs and Dimmito, Marilisa Pia and Sebastiani, Jessica and La Regina, Giuseppe and Silvestri, Romano and Tömböly, Csaba (2023) Rimonabant-Based Compounds Bearing Hydrophobic Amino Acid Derivatives as Cannabinoid Receptor Subtype 1 Ligands. ACS MEDICINAL CHEMISTRY LETTERS, 14 (4). pp. 479-486. ISSN 1948-5875

Szabó, Renáta and Szabó, Zsuzsanna and Börzsei, Denise and Nagyné Hoffmann, Alexandra and Lesi, Zelma Nadin and Pálszabó, Patrícia and Pálszabó, Andrea and Dvorácskó, Szabolcs and Gesztelyi, Rudolf and Kupai, Krisztina and Priksz, Dániel and Juhász, Béla and Altmayer, Anita and Varga, Csaba and Pósa, Anikó (2022) Potential Implications of Rimonabant on Age-Related Oxidative Stress and Inflammation. ANTIOXIDANTS, 11 (1). pp. 1-14. ISSN 2076-3921

Almási, Nikoletta and Murlasits, Z. and Al-Awar, Amin and Csonka, Ákos and Dvorácskó, Szabolcs and Tömböly, Csaba and Török, Szilvia and Pósa, Anikó and Varga, Csaba and Kupai, Krisztina (2021) Effects of aging on proteasomal-ubiquitin system, oxidative stress balance and calcium homeostasis in middle-aged female rat colon. Physiology International, 108 (1). pp. 27-42. ISSN 2498-602X

Szabó, Írisz and Varga, Viktória É. and Dvorácskó, Szabolcs and Farkas, Elek Attila and Körmöczi, Tímea and Berkecz, Róbert and Kecskés, Szilvia and Menyhárt, Ákos and Frank, Rita and Frecska, Ede and Tömböly, Csaba and Krizbai, István Adorján and Bari, Ferenc and Farkas, Eszter (2021) N,N-Dimethyltryptamine attenuates spreading depolarization and restrains neurodegeneration by sigma-1 receptor activation in the ischemic rat brain. NEUROPHARMACOLOGY, 192. ISSN 0028-3908

Dvorácskó, Szabolcs and Lázár, László and Fülöp, Ferenc and Palkó, Márta and Zalán, Zita and Penke, Botond and Fülöp, Lívia and Tömböly, Csaba and Bogár, Ferenc (2021) Novel High Affinity Sigma-1 Receptor Ligands from Minimal Ensemble Docking-Based Virtual Screening. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 22 (15). pp. 1-17. ISSN 1661-6596 (print); 1422-0067 (online)

Zádor, Ferenc and Joca, Sâmia and Nagy-Grócz, Gábor and Dvorácskó, Szabolcs and Szűcs, Edina and Tömböly, Csaba and Benyhe, Sándor and Vécsei, László (2021) Pro-Inflammatory Cytokines: Potential Links between the Endocannabinoid System and the Kynurenine Pathway in Depression. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 22 (11). ISSN 1661-6596

Almási, Nikoletta and Török, Szilvia and Dvorácskó, Szabolcs and Tömböly, Csaba and Csonka, Ákos and Baráth, Zoltán Lajos and Murlasits, Zsolt and Valkusz, Zsuzsanna and Pósa, Anikó and Varga, Csaba and Kupai, Krisztina (2020) Lessons on the Sigma-1 Receptor in TNBS-Induced Rat Colitis. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 21 (11). ISSN 1661-6596

Zádor, Ferenc and Nagy-Grócz, Gábor and Dvorácskó, Szabolcs and Bohár, Zsuzsanna and Cseh, Edina Katalin and Zádori, Dénes and Párdutz, Árpád and Szűcs, Edina and Tömböly, Csaba and Borsodi, Anna and Benyhe, Sándor and Vécsei, László (2020) Long-term systemic administration of kynurenic acid brain region specifically elevates the abundance of functional CB1 receptors in rats. NEUROCHEMISTRY INTERNATIONAL, 138. ISSN 0197-0186

Dimmito, Marilisa P. and Stefanucci, Azzurra and Pieretti, Stefano and Minosi, Paola and Dvorácskó, Szabolcs and Tömböly, Csaba and Zengin, Gokhan and Mollica, Adriano (2019) Discovery of Orexant and Anorexant Agents with Indazole Scaffold Endowed with Peripheral Antiedema Activity. BIOMOLECULES, 9 (9). ISSN 2218-273X

Zádor, Ferenc and Nagy-Grócz, Gábor and Kékesi, Gabriella and Dvorácskó, Szabolcs and Szűcs, Edina and Tömböly, Csaba and Horváth, Gyöngyi and Benyhe, Sándor and Vécsei, László (2019) Kynurenines and the Endocannabinoid System in Schizophrenia: Common Points and Potential Interactions. MOLECULES, 24 (20). pp. 1-36. ISSN 1420-3049

Dvorácskó, Szabolcs and Keresztes, Attila and Mollica, Adriano and Stefanucci, Azzurra and Macedonio, Giorgia and Zádor, Ferenc and Walter, Fruzsina R. and Deli, Mária A. and Kékesi, Gabriella and Bánki, László and Tuboly, Gábor and Horváth, Gyöngyi and Tömböly, Csaba (2019) Preparation of bivalent agonists for targeting the mu opioid and cannabinoid receptors. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 178. pp. 571-588. ISSN 0223-5234

Stefanucci, Azzurra and Novellino, Ettore and Macedonio, Giorgia and Dimmito, Marilisa Pia and Mirzaie, Sako and Cardoso, Fernanda Caldas and Lewis, Richard and Zádor, Ferenc and Erdei, Anna and Dvorácskó, Szabolcs and Tömböly, Csaba and Benyhe, Sándor and Pieretti, Stefano and Minosi, Paola and Mollica, Adriano (2018) Design, synthesis and biological profile of mixed opioid agonist/N-VGCC blocker peptides. NEW JOURNAL OF CHEMISTRY, 42 (8). pp. 5656-5659. ISSN 1144-0546

Leone, Sheila and Ferrante, Claudio and Recinella, Lucia and Chiavaroli, Annalisa and Mollica, Adriano and Tömböly, Csaba and Stefanucci, Azzurra and Dimmito, Marilisa Pia and Dvorácskó, Szabolcs and Verratti, Vittore and De Petrocellis, Luciano and Orlando, Giustino and Brunetti, Luigi (2018) Effects of RVD-hemopressin (α) on feeding and body weight after standard or cafeteria diet in rats. NEUROPEPTIDES, 72. pp. 38-46. ISSN 0143-4179

Stefanucci, Azzurra and Macedonio, Giorgia and Dvorácskó, Szabolcs and Tömböly, Csaba and Mollica, Adriano (2018) Novel Fubinaca/Rimonabant hybrids as endocannabinoid system modulators. AMINO ACIDS, 50 (11). pp. 1595-1605. ISSN 0939-4451

Mollica, A. and Pelliccia, S. and Famiglini, V. and Stefanucci, A. and Macedonio, G. and Benyhe, Sándor and Zádor, Ferenc and Erdei, Anna and Szűcs, Edina and Samavati, Reza and Dvorácskó, Szabolcs and Tömböly, Csaba (2017) Exploring the first Rimonabant analog-opioid peptide hybrid compound, as bivalent ligand for CB1 and opioid receptors. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 32 (1). pp. 444-451. ISSN 1475-6366

Adamska-Bartlomiejczyk, Anna and Borics, Attila and Tömböly, Csaba and Dvorácskó, Szabolcs and Lisowski, Marek (2017) Synthesis, receptor binding studies, optical spectroscopic and in silico structural characterization of morphiceptin analogs with cis-4-amino-L-proline residues. JOURNAL OF PEPTIDE SCIENCE, 23 (12). pp. 864-870. ISSN 1075-2617

Szűcs, Edina and Dvorácskó, Szabolcs and Tömböly, Csaba and Büki, Alexandra and Kékesi, Gabriella and Horváth, Gyöngyi and Benyhe, Sándor (2016) Decreased CB receptor binding and cannabinoid signaling in three brain regions of a rat model of schizophrenia. NEUROSCIENCE LETTERS, 633. pp. 87-93. ISSN 0304-3940

Monti, L. and Stefanucci, A. and Pieretti, S. and Marzoli, F. and Fidanza, L. and Benyhe, Sándor and Zádor, Ferenc and Szűcs, Edina and Ötvös, Ferenc and Erdei, Anna and Samavati, Reza and Dvorácskó, Szabolcs and Tömböly, Csaba (2016) Evaluation of the analgesic effect of 4-anilidopiperidine scaffold containing ureas and carbamates. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 31 (6). pp. 1638-1647. ISSN 1475-6366

Mollica, Adriano and Mirzaie, Sarra and Costante, Roberto and Carradori, Simone and Macedonio, G. and Dvorácskó, Szabolcs (2016) Exploring the biological consequences of conformational changes in aspartame models containing constrained analogues of phenylalanine. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 31 (6). pp. 953-963. ISSN 1475-6366

Dvorácskó, Szabolcs and Tömböly, Csaba and Berkecz, Róbert and Keresztes, Attila (2016) Investigation of receptor binding and functional characteristics of hemopressin(1-7). NEUROPEPTIDES, 58. pp. 15-22. ISSN 0143-4179

Dvorácskó, Szabolcs and Stefanucci, Azzurra and Novellino, Ettore and Mollica, Adriano (2015) The design of multitarget ligands for chronic and neuropathic pain. Future Medicinal Chemistry, 7 (18). pp. 2469-2483. ISSN 1756-8919

This list was generated on Tue Dec 9 15:13:41 2025 CET.