Items where Author is "Schneider, Gyula"

Article

Kiss, Anita and Jójárt, Rebeka and Mernyák, Erzsébet and Bartha, Sándor and Minorics, Renáta and Zupkó, István and Schneider, Gyula (2021) Novel preparation of substituted oxazolines condensed to d-ring of estrane skeleton and characterization of their antiproliferative properties. STEROIDS. ISSN 0039-128X (In Press)

Nagymihály, Zoltán and Wölfling, János and Schneider, Gyula and Kollár, László (2020) Synthesis of 2-Methylresorcinol-Based Deepened Cavitands with Chiral Inlet Bearing Steroidal Moieties on the Upper Rim. ChemistrySelect. pp. 6933-6938. ISSN 2365-6549

Herman, Bianka Edina and Kiss, Anita and Wölfling, János and Mernyák, Erzsébet and Szécsi, Mihály and Schneider, Gyula (2019) Synthesis of substituted 15β-alkoxy estrone derivatives and their cofactor-dependent inhibitory effect on 17β-HSD1. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 34 (1). pp. 1271-1286. ISSN 1475-6366

Jójárt, Rebeka and Traj, Péter and Kovács, Édua and Horváth, Ágnes and Schneider, Gyula and Szécsi, Mihály and Pál, Attila and Paragi, Gábor and Mernyák, Erzsébet (2019) Synthesis, Biological Evaluation and Docking Studies of 13-Epimeric 10-fluoro- and 10-Chloroestra-1,4-dien-3-ones as Potential Aromatase Inhibitors. MOLECULES, 24 (9). No.-1783. ISSN 1420-3049

Bacsa, Ildikó and Szemerédi, Dávid and Wölfling, János and Schneider, Gyula and Fekete, Lilla and Mernyák, Erzsébet (2018) The first Pd-catalyzed Buchwald–Hartwig aminations at C-2 or C-4 in the estrone series. BEILSTEIN JOURNAL OF ORGANIC CHEMISTRY. ISSN 1860-5397

Gyovai, András and Minorics, Renáta and Kiss, Anita and Mernyák, Erzsébet and Schneider, Gyula and Szekeres, András and Kerekes, Erika and Ocsovszki, Imre and Zupkó, István (2018) Antiproliferative Properties of Newly Synthesized 19-Nortestosterone Analogs Without Substantial Androgenic Activity. FRONTIERS IN PHARMACOLOGY, 9. pp. 1-11. ISSN 1663-9812

Bacsa, Ildikó and Herman, Bianka Edina and Jójárt, Rebeka and Herman, Kevin Stefán and Wölfling, János and Schneider, Gyula and Varga, Mónika and Tömböly, Csaba and Szécsi, Mihály and Mernyák, Erzsébet (2018) Synthesis and structure–activity relationships of 2- and/or 4-halogenated 13β- and 13α-estrone derivatives as enzyme inhibitors of estrogen biosynthesis. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 33 (1). pp. 1271-1282. ISSN 1475-6366 (print); 1475-6374 (online)

Fröhlich, Tony and Kiss, Anita and Wölfling, János and Mernyák, Erzsébet and Kulmány, Ágnes E. and Minorics, Renáta and Zupkó, István and Schneider, Gyula (2018) Synthesis of Artemisinin-Estrogen Hybrids Highly Active against HCMV, P. falciparum, and Cervical and Breast Cancer. ACS MEDICINAL CHEMISTRY LETTERS, 9 (11). pp. 1-6. ISSN 1948-5875

Bózsity, Noémi and Minorics, Renáta and Szabó, Johanna and Mernyák, Erzsébet and Schneider, Gyula and Wölfling, János and Ocsovszki, Imre and Zupkó, István (2017) Mechanism of antiproliferative action of a new D-secoestrone-triazole derivative in cervical cancer cells and its effect on cancer cell motility. JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 165. pp. 247-257. ISSN 0960-0760

Bacsa, Ildikó and Jójárt, Rebeka and Wölfling, János and Schneider, Gyula and Herman, Bianka Edina and Szécsi, Mihály and Mernyák, Erzsébet (2017) Synthesis of novel 13 α-estrone derivatives by Sonogashira coupling as potential 17 β-HSD1 inhibitors. BEILSTEIN JOURNAL OF ORGANIC CHEMISTRY, 13. pp. 1303-1309. ISSN 1860-5397

Bózsity, Noémi and Minorics, Renáta and Szabó, Johanna and Mernyák, Erzsébet and Schneider, Gyula and Wölfling, János and Wang, Hui-Chun and Wu, Chin-Chung and Ocsovszki, Imre and Zupkó, István (2016) Mechanism of antiproliferative action of a new D-secoestrone-triazole derivative in cervical cancer cells and its effect on cancer cell motility. JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY. ISSN 0960-0760 (In Press)

Schneider, Gyula and Kiss, Anita and Mernyák, Erzsébet and Benke, Zsanett and Wölfling, János and Frank, Éva and Bózsity, Noémi and Gyovai, András and Minorics, Renáta and Zupkó, István (2016) Stereocontrolled synthesis of the four 16-hydroxymethyl-19- nortestosterone isomers and their antiproliferative activities. STEROIDS, 105. pp. 113-120. ISSN 0039-128X

Schneider, Gyula and Kiss, Anita and Mernyák, Erzsébet and Benke, Zsanett and Wölfling, János and Frank, Éva and Bózsity, Noémi and Gyovai, András and Minorics, Renáta and Zupkó, István (2016) Stereocontrolled synthesis of the four 16-hydroxymethyl-19-nortestosterone isomers and their antiproliferative activities. STEROIDS, 105. pp. 113-120. ISSN 0039-128X

Szabó, Johanna and Pataki, Zoltán and Wölfling, János and Schneider, Gyula and Bózsity, Noémi and Minorics, Renáta and Zupkó, István and Mernyák, Erzsébet (2016) Synthesis and biological evaluation of 13a-estrone derivatives as potential antiproliferative agents. STEROIDS, 113. pp. 14-21. ISSN 0039-128X

Szabó, Johanna and Pataki, Zoltán and Wölfling, János and Schneider, Gyula and Bózsity, Noémi and Minorics, Renáta and Zupkó, István and Mernyák, Erzsébet (2016) Synthesis and biological evaluation of 13α-estrone derivatives as potential antiproliferative agents. STEROIDS, 113. pp. 14-21. ISSN 0039-128X

Szabó, Johanna and Jerkovics, Nóra and Schneider, Gyula and Wölfling, János and Bózsity, Noémi and Minorics, Renáta and Zupkó, István and Mernyák, Erzsébet (2016) Synthesis and in Vitro Antiproliferative Evaluation of C-13 Epimers of Triazolyl-D-Secoestrone Alcohols: The First Potent 13α-D-Secoestrone Derivative. MOLECULES, 21 (611). ISSN 1420-3049

Szabó, Johanna and Jerkovics, Nóra and Schneider, Gyula and Wölfling, János and Bózsity, Noémi and Minorics, Renáta and Zupkó, István and Mernyák, Erzsébet (2016) Synthesis and in Vitro Antiproliferative Evaluation of C-13 Epimers of Triazolyl-D-Secoestrone Alcohols: The First Potent 13α-D-Secoestrone Derivative. MOLECULES, 21 (5). pp. 1-13. ISSN 1420-3049

Mótyán, Gergő and Zupkó, István and Minorics, Renáta and Schneider, Gyula and Wölfling, János and Frank, Éva (2015) Lewis acid-induced intramolecular access to novel steroidal ring D-condensed arylpyrazolines exerting in vitro cell-growth-inhibitory effects. MOLECULAR DIVERSITY .

Szabó, Nikoletta and Iványi, Zoltán and Szécsi, Mihály and Julesz, János and Mernyák, Erzsébet and Huber, Judit and Wölfling, János and Minorics, Renáta and Zupkó, István and Schneider, Gyula (2015) Synthesis of methoxycarbonylpyrazolylandrostene derivatives, and their potential inhibitory effect on androgen biosynthesis and cell proliferation. STEROIDS, 98. pp. 143-152. ISSN 0039-128X

Schneider, Gyula and Görbe, Tamás and Mernyák, Erzsébet and Wölfling, János and Holczbauer, Tamás and Minorics, Renáta and Zupkó, István (2015) Synthesis of novel 17-(5’-iodo)triazolyl-3-methoxyestrane epimers via Cu(I)-catalyzed azide-alkyne cycloadditon, and an evaluation of their cytotoxic activity in vitro. STEROIDS, 98. pp. 153-165. ISSN 0039-128X

Mernyák, Erzsébet and Kovács, Ida and Minorics, Renáta and Sere, Péter and Czégány, Dóra and Wölfling, János and Schneider, Gyula and Újfaludi, Zsuzsanna and Boros, Imre Miklós and Zupkó, István (2015) Synthesis of trans-16-triazolyl-13α-methyl-17-estradiol diastereomers and the effects of structural modifications on their in vitro antiproliferative activities. JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 150. pp. 123-134. ISSN 0960-0760

Iványi, Zoltán and Görbe, Tamás and Szabó, Nikoletta and Kiss, Anita and Wölfling, János and Schneider, Gyula (2014) 17ß-Pirazolil- és -pirazolinil-szteroidok szintézise. MAGYAR KÉMIAI FOLYÓIRAT - KÉMIAI KÖZLEMÉNYEK, 120 (2-3). pp. 116-121. ISSN 1418-9933

Schneider, Gyula and Matkovics, Béla and Zsolt, János (1960) Néhány adat a difenilamin karotinoidszintézisre gyakorolt hatására vonatkozóan. A MAGYAR TUDOMÁNYOS AKADÉMIA BIOLÓGIAI CSOPORTJÁNAK KÖZLEMÉNYEI, 4 (3-4). pp. 281-285.

Monograph

Schneider, Gyula and Nagyné dr. Frank, Éva and Wölfling, János (2011) Szteránvázas vegyületek kutatása = Research of steroids. Project Report. OTKA.

Wölfling, János and Julesz, János and Mernyák, Erzsébet and Nagyné dr. Frank, Éva and Schneider, Gyula and Szájli, Ágota and Szécsi, Mihály and Tóth, István (2009) Antiandrogén kardenolid analógok szintézise és biológiai hatásvizsgálata = Synthesis and biological effect investigations of antiandrogen cardenolide analogues. Project Report. OTKA.

Schneider, Gyula and Magyar, Angéla Andrea and Mernyák, Erzsébet and Nagyné dr. Frank, Éva and Wölfling, János (2007) Szteránvázas vegyületek szintézise = Synthesis of Steroid Compounds. Project Report. OTKA.